Esomeprazole Magnesium Capsules (esomeprazole ... | 合法藥品大搜索
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EsomeprazoleMagnesiumisaprescriptionandover-the-countermedicineusedtotreatthesymptomsofheartburn,GERDwithorwithoutErosiveEsophagitis, ...
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Esomeprazole is a proton pump inhibitor that suppresses gastric acid secretion by specific inhibition of the H+/K+-ATPase in the gastric parietal[1] cell. The S- and R-isomers of omeprazole are protonated and converted in the acidic compartment of the parietal cell forming the active inhibitor, the achiral sulphenamide. By acting specifically on the proton pump, esomeprazole blocks the final step in acid production, thus reducing gastric acidity. This effect is dose-related up to a daily dose of 20 mg to 40 mg and leads to inhibition of gastric acid secretion.
Pharmacodynamics Antisecretory ActivityThe effect of esomeprazole magnesium delayed-release capsules on intragastric pH was determined in patients with symptomatic gastroesophageal[2] reflux[3] disease in two separate studies. In the first study of 36 patients...
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