[Vasopressin receptor antagonists | 合法藥品大搜索
![[Vasopressin receptor antagonists](https://i.imgur.com/IMDjKGl.jpg)
由CVillabona著作·2010·被引用6次—Thenon-peptidevasopressinantagonists(VPA),calledvaptans,weredevelopedinthe1990stoantagonizeboththepressorandantidiureticeffectsof ...
![[Vasopressin receptor antagonists](https://i.imgur.com/IMDjKGl.jpg)
The non-peptide vasopressin antagonists (VPA), called vaptans, were developed in the 1990s to antagonize both the pressor and antidiuretic effects of vasopressin. There are three subtypes of VPA receptors: V1a, V1b and V2. V1a receptors are widely distributed in the body, mainly the blood vessels and myocardium. The V1b receptors are located mainly in the anterior pituitary gland and play a role in ACTH release. V2 receptors are located in the collecting tubular renal cells. Both V1a and V1b receptors act through the intracellular phosphoinositol signalling pathway, Ca(++) being the second messenger. V2 receptors work through AMPc generation, which promotes aquaporin 2 (AQP2) trafficking and allows water to enter the cell. The vaptans act competitively at the AVP receptor. The most important are mozavaptan, lixivaptan, satavaptan and tolvaptan, all of which are selective V2 antagonists and are administered through t...
Clinical review | 合法藥品大搜索
Non-peptide arginine | 合法藥品大搜索
Vaptans for the treatment of hyponatremia | 合法藥品大搜索
Vaptans for the treatment of hyponatremia | 合法藥品大搜索
Vaptans | 合法藥品大搜索
Vaptans | 合法藥品大搜索
Vasopressin receptor antagonist | 合法藥品大搜索
[Vasopressin receptor antagonists | 合法藥品大搜索
“Tolvaptan”一種專一性vasopressin | 合法藥品大搜索
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