Epileptogenic Potential of Carbapenem Agents | 合法藥品大搜索
KeyWords:carbapenem,imipenem,meropenem,doripenem,ertapenem,seizure,epilepsy...mechanismsfordrug-inducedseizure,riskfactors,anddrug ...
Antimicrobials are the most frequently implicated class of drugs in drug-induced seizure, with β-lactams being the class of antimicrobials most often implicated. The seizure-inducing potential of the carbapenem subclass may be directly related to their β-lactam ring structure. Data on individual carbapenems and seizure activity are scarce. To evaluate the available evidence on the association between carbapenem agents and seizure activity, we conducted a literature search of the MEDLINE (1966—May 2010), EMBASE (1974–May 2010), and International Pharmaceutical Abstracts (1970—May 2010) databases. Reference citations from the retrieved articles were also reviewed. Mechanistically, seizure propensity of the β-lactams is related to their binding to 7-aminobutyric acid (GABA) receptors. There are numerous reports of seizure activity associated with imipenem-cilastatin, with seizure rates ranging from 3–33%. For meropenem, doripenem, and ertapenem, the seizure rate for each agen...
Risk factors associated with the development of ... | 合法藥品大搜索
The risk of seizures among the carbapenems | 合法藥品大搜索
Epileptogenic potential of carbapenem agents ... | 合法藥品大搜索
Risk factors associated with the development of ... | 合法藥品大搜索
The risk of seizures among the carbapenems | 合法藥品大搜索
Status Epilepticus and Delirium Associated with Ertapenem in ... | 合法藥品大搜索
risk of seizures among the carbapenems | 合法藥品大搜索
Higher than expected rates of seizures associated with the ... | 合法藥品大搜索
Epileptogenic Potential of Carbapenem Agents | 合法藥品大搜索
Seizures associated with ertapenem use in patients with CNS ... | 合法藥品大搜索
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